Sairam V. V. M. Kalapatapu

Employment

Employment history is unavailable.

Education

Education history is unavailable.

Projects & Funding

Projects & funding information is unavailable.

Publications (20)

• In the Quest for Potent and Selective Malic Enzyme 3 Inhibitors for the Treatment of Pancreatic Ductal Adenocarcinoma
  ACS Medicinal Chemistry Letters 2023 DOI: 10.1021/acsmedchemlett.2c00369
  +Save
• Discovery of a Potent and Orally Efficacious TGR5 Receptor Agonist
  ACS Medicinal Chemistry Letters 2016 DOI: 10.1021/acsmedchemlett.5b00323
  +Save
• Design, synthesis and biological evaluation of novel aminomethyl-piperidones based DPP-IV inhibitors
  Bioorganic & Medicinal Chemistry Letters 2014 DOI: 10.1016/j.bmcl.2014.03.009
  +Save
• Peptidomimetics as Potent and Selective PTP1B Inhibitors
  Medicinal Chemistry 2013 DOI: 10.2174/1573406411309050005
  +Save
• Synthesis and structure–activity relationship of potent, selective and orally active anthranilamide-based factor Xa inhibitors: Application of weakly basic sulfoximine group as novel S4 binding element
  European Journal of Medicinal Chemistry 2012 DOI: 10.1016/j.ejmech.2012.10.005
  +Save
• Design of Peptidomimetic Based DPP-IV Inhibitors, Devoid of CYP Liabilities
  Letters in Drug Design & Discovery 2012 DOI: 10.2174/157018012803307932
  +Save
• Discovery of liver selective non-steroidal glucocorticoid receptor antagonist as novel antidiabetic agents
  Bioorganic & Medicinal Chemistry Letters 2012 DOI: 10.1016/j.bmcl.2012.07.078
  +Save
• Long-acting peptidomimetics based DPP-IV inhibitors
  Bioorganic & Medicinal Chemistry Letters 2012 DOI: 10.1016/j.bmcl.2012.03.078
  +Save
• Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors
  Bioorganic & Medicinal Chemistry Letters 2012 DOI: 10.1016/j.bmcl.2011.11.122
  +Save
• Discovery of Orally Active, Potent, and Selective Benzotriazole-Based PTP1B Inhibitors
  ChemMedChem 2011 DOI: 10.1002/cmdc.201100077
  +Save