Kalpana Tilekar

Employment

• Bharati Vidyapeeth's College of Pharmacy Assistant Professor
  2021 - Present
• Bharati Vidyapeeth's College of Pharmacy PhD student & Research Fellow
  2017 - 2021

Education

Education history is unavailable.

Projects & Funding

Projects & funding information is unavailable.

Publications (14)

• Synthesis, In‐Vitro Evaluation and Molecular Docking Study of N‐Substituted Thiazolidinediones as α‐Glucosidase Inhibitors
  ChemistrySelect 2022 DOI: 10.1002/slct.202103848
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• Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4
  Pharmaceuticals 2021 DOI: 10.3390/ph14101032
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• Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy
  Bioorganic Chemistry 2021 DOI: 10.1016/j.bioorg.2020.104527
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• Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential
  European Journal of Medicinal Chemistry 2020 DOI: 10.1016/j.ejmech.2020.112603
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• Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib
  Bioorganic and Medicinal Chemistry Letters 2020 DOI: 10.1016/j.bmcl.2020.127561
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• Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines
  Bioorganic Chemistry 2020 DOI: 10.1016/j.bioorg.2019.103522
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• Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation
  Bioorganic Chemistry 2020 DOI: 10.1016/j.bioorg.2020.103934
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• Permuted 2,4-thiazolidinedione (TZD) analogs as GLUT inhibitors and their in-vitro evaluation in leukemic cells
  European Journal of Pharmaceutical Sciences 2020 DOI: 10.1016/j.ejps.2020.105512
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• Power of two: combination of therapeutic approaches involving glucose transporter (GLUT) inhibitors to combat cancer
  Biochimica et Biophysica Acta - Reviews on Cancer 2020 DOI: 10.1016/j.bbcan.2020.188457
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• Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents
  ChemMedChem 2020 DOI: 10.1002/cmdc.202000458
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