Nilesh Khedkar

Employment

• Lupin Ltd Research and Development Scientist
  2011 - Present
• Zydus Research Center Chemist
  2008 - 2011

Education

Education history is unavailable.

Projects & Funding

Projects & funding information is unavailable.

Publications (5)

• Computational Design, Synthesis, and Bioevaluation of 2-(Pyrimidin-4-yl)oxazole-4-carboxamide Derivatives: Dual Inhibition of EGFRWT and EGFRT790M with ADMET Profiling
  Bioorganic Chemistry 2024 DOI: 10.1016/j.bioorg.2023.107027
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• Computational design, synthesis, and assessment of 3-(4-(4-(1,3,4-oxadiazol-2-yl)-1H-imidazol-2-yl)phenyl)-1,2,4-oxadiazole derivatives as effective epidermal growth factor receptor inhibitors: a prospective strategy for anticancer therapy
  RSC Medicinal Chemistry 2024 DOI: 10.1039/d4md00055b
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• Design, synthesis, and characterization of 3-(2-(pyrimidin-5-yl)thiazol-4-yl)-1,2,4-oxadiazole derivatives: Anticancer and molecular docking investigations
  Synthetic Communications 2023 DOI: 10.1080/00397911.2023.2287796
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• Discovery of a Novel Potent and Selective Calcium Release-Activated Calcium Channel Inhibitor: 2,6-Difluoro- N-(2′-methyl-3′-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1′-biphenyl]-4-yl)benzamide. Structure-Activity Relationship and Preclinical…
  Journal of Medicinal Chemistry 2021 DOI: 10.1021/acs.jmedchem.1c01403
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• Discovery of isoquinolinone and naphthyridinone-based inhibitors of poly(ADP-ribose) polymerase-1 (PARP1) as anticancer agents: Structure activity relationship and preclinical characterization
  Bioorganic and Medicinal Chemistry 2020 DOI: 10.1016/j.bmc.2020.115819
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