Prabhakar Koiram Rajanna

Employment

• Bristol-Myers Squibb Co Research & Development Lead Investigator & Functional head
  2021 - Present
• Biocon Bristol-Myers Squibb Research and Development Center Senior Prinicpal Investigator
  2014 - 2021
• AstraZeneca India Private Limited Research Scientist 2
  2012 - 2014
• Advinus Therapeutics Private Limited Senior Research Scientist
  2008 - 2012
• Ecron Acunova Research Scientist
  2007 - 2008
• Himalaya Drug Company Research Executive
  2002 - 2004
• Sri KV College of Pharmacy Lecturer
  2000 - 2002

Education

• Manipal University PhD
  2004 - 2007
• Manipal College of Pharmaceutical Sciences M Pharm
  2000 - 2002
• PES College of Pharmacy
  1994 - 1997

Projects & Funding

Projects & funding information is unavailable.

Publications (49)

• Discovery of Imidazopyridines as Potent Inhibitors of Indoleamine 2,3-Dioxygenase 1 for Cancer Immunotherapy.
  ACS medicinal chemistry letters 2021 12 citations DOI: 10.1021/acsmedchemlett.1c00014
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• Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors.
  ACS medicinal chemistry letters 2021 5 citations DOI: 10.1021/acsmedchemlett.1c00236
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• U.S. FDA Approved Drugs from 2015-June 2020: A Perspective.
  Journal of medicinal chemistry 2021 790 citations DOI: 10.1021/acs.jmedchem.0c01786
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• Qualified method for the estimation of di-18:1 bis(monoacylglycero)phosphate in urine, a noninvasive biomarker to monitor drug-induced phospholipidosis.
  Bioanalysis 2020 2 citations DOI: 10.4155/bio-2020-0114
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• Impact of quercetin on pharmacokinetics of quetiapine: insights from in-vivo studies in wistar rats.
  Xenobiotica; the fate of foreign compounds in biological systems 2020 6 citations DOI: 10.1080/00498254.2020.1792002
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• Is aspirin a substrate of MDR1/P-glycoprotein?
  Xenobiotica; the fate of foreign compounds in biological systems 2020 2 citations DOI: 10.1080/00498254.2020.1757785
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• Evidence for the Validity of Pyridoxic Acid (PDA) as a Plasma-Based Endogenous Probe for OAT1 and OAT3 Function in Healthy Subjects.
  The Journal of pharmacology and experimental therapeutics 2018 59 citations DOI: 10.1124/jpet.118.252643
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• Offline derivatization LC-MS/MS method for simultaneous estimation of vanillin and vanillic acid in guinea pig plasma.
  Bioanalysis 2018 9 citations DOI: 10.4155/bio-2017-0213
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• Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis.
  Journal of medicinal chemistry 2017 126 citations DOI: 10.1021/acs.jmedchem.6b01358
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• Enantioselective supercritical fluid chromatography–tandem mass spectrometry method for simultaneous estimation of risperidone and its 9-hydroxyl metabolites in rat plasma
  Bioanalysis 2017 13 citations DOI: 10.4155/bio-2017-0168
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